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14

抑制剂 & 化合物

3

天然产物

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Cat. No. Product Name Target Signaling Pathways
T1444 Lomefloxacin

洛美沙星,SC47111A

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Lomefloxacin (SC47111A) 是一种广谱喹诺酮类抗生素,具有抗菌活性。它可研究支气管炎、尿路感染、结膜炎、外耳炎和中耳炎。
T1070 Cefmetazole sodium

头孢美唑钠,Sodium cefmetazole

Antibacterial; Antibiotic Microbiology/Virology
Cefmetazole sodium (Sodium cefmetazole) 是具有广谱抗菌活性的半合成头孢霉素抗生素。它通过与青霉素结合蛋白结合,阻止肽聚糖的交联,导致细胞壁完整性的丧失。它可研究妇科、腹腔内、尿道、呼吸道和皮肤和软组织感染。
T0748 Sulfameter

5-Methoxysulfadiazine,Sulfametoxydiazine,磺胺对甲氧嘧啶

DHFR; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Sulfameter (Sulfametoxydiazine) 是一种长效磺胺类抗生素,具有抗菌活性。它可研究尿路感染和麻风病。
T6349 Sitafloxacin Hydrate

西他沙星水合物,DU-6859a,DU6859a hydrate

Antibacterial; Antibiotic Microbiology/Virology
Sitafloxacin Hydrate (DU-6859a) 是一种口服有效的氟喹诺酮类抗生素,在体外可对抗广泛的革兰氏阳性和阴性细菌有活性。Sitafloxacin 可研究呼吸道感染和尿路感染。
T8139 Sulfamethoxazole sodium

新诺明钠,Ro 4-2130 sodium,磺胺甲恶唑钠

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Sulfamethoxazole sodium (Ro 4-2130 sodium) 是一种磺胺类抗菌素。它常用于各种尿道病原体的研究,与 Trimethoprim 联用,可用于尿路感染的研究。
T1625 Lomefloxacin hydrochloride

Lomefloxacin HCl,盐酸洛美沙星,Okacyn,Maxaquin

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Lomefloxacin hydrochloride (Okacyn) 是一种广谱喹诺酮类抗生素,具有抗菌活性。它可研究支气管炎、尿路感染、结膜炎、外耳炎和中耳炎。
T8722 iKIX1

Antifungal Microbiology/Virology
iKIX1 是一种 Pdr1 依赖性基因激活。 它在体外和在播散性和泌尿道光滑念珠菌感染的动物模型中使耐药的光滑念珠菌对唑类抗真菌剂重新敏感。它可研究多药耐药性和光滑念珠菌感染。
T30737 Carbavance

Meropenem/vaborbactam,Vabomere

Carbavance, a mixture of Meropenham and Vaborbactam, is intended for adults with complex urinary tract infections (cUTI), including pyelonephritis, a kidney infection caused by certain bacteria.
T40295 Carindacillin sodium

Carindacillin sodium,CP-15464-2,Carbenicillin indanyl sodium

Carindacillin sodium, also known as Carbenicillin indanyl sodium, is an orally active, broad-spectrum antimicrobial agent. In vivo, it undergoes hydrolysis to Carbenicillin. Carindacillin sodium is specifically utilized in urinary tract infection research.
T34776 Talampicillin

Talampicillin is an ester of Ampicillin. It is hydrolyzed upon absorption to release ampicillin. It is well absorbed from the gastrointestinal tract resulting in a greater bioavailability of ampicillin than can be achieved with equivalent doses of ampicil
T36537 Nitrofurantoin-13C3

Nitrofurantoin-13C3

Nitrofurantoin-13C3is intended for use as an internal standard for the quantification of nitrofurantoin by GC- or LC-MS. Nitrofurantoin is a nitrofuran antibiotic.1In vivo, nitrofurantoin (25-100 mg/kg) reducesE. colireplication and abscess formation in the renal medulla of infected rats in a dose-dependent manner. It prevents kidney and bladder infection in rats following bladder inoculation with clinical isolates ofP. mirabilis. Nitrofurantoin also prevents alkalization of urine, as well as ca...
T75291 Trimethoprim hydrochloride

Trimethoprim hydrochloride 是一种口服活性的抑菌抗生素,同时也是二氢叶酸还原酶抑制剂。它对多种革兰氏阳性及革兰氏阴性需氧细菌有效。用于尿路感染、志贺氏菌病和肺孢子菌肺炎的研究。与锌联合使用时,可抑制甲型流感病毒对鸡胚的感染。
T36021 Flumequine-13C3

Flumequine-13C3

Flumequine-13C3is intended for use as an internal standard for the quantification of flumequine by GC- or LC-MS. Flumequine is a fluoroquinolone antibiotic.1It is active againstS. aureus, S. pyogenes, B. subtilis, E. coli, P. aeruginosa, S. faecalis, andK. pneumoniae(MICs = 1-100 μg/ml). Flumequine is also active against field isolates of B. hyodysenteriae (MICs = 6.25-200 μg/ml).2It inhibits DNA gyrase, disrupting supercoiling of bacterial DNA to block transcription and replication.3In vivo, fl...
T75296 Pazufloxacin

Pazufloxacin (T-3761)是氟喹诺酮类广谱抗生素。

化合物

Lomefloxacin
Cat.No: T1444
Synonym: 洛美沙星,SC47111A
Target: Topoisomerase, Antibacterial, Antibiotic
Cefmetazole sodium
Cat.No: T1070
Synonym: 头孢美唑钠,Sodium cefmetazole
Target: Antibacterial, Antibiotic
Sulfameter
Cat.No: T0748
Synonym: 5-Methoxysulfadiazine,Sulfametoxydiazine,磺胺对甲氧嘧啶
Target: DHFR, Antibacterial, Antibiotic
Sitafloxacin Hydrate
Cat.No: T6349
Synonym: 西他沙星水合物,DU-6859a,DU6859a hydrate
Target: Antibacterial, Antibiotic
Sulfamethoxazole sodium
Cat.No: T8139
Synonym: 新诺明钠,Ro 4-2130 sodium,磺胺甲恶唑钠
Target: Others, Antibacterial, Antibiotic
Lomefloxacin hydrochloride
Cat.No: T1625
Synonym: Lomefloxacin HCl,盐酸洛美沙星,Okacyn,Maxaquin
Target: Topoisomerase, Antibacterial, Antibiotic
iKIX1
Cat.No: T8722
Synonym:
Target: Antifungal
Carbavance
Cat.No: T30737
Synonym: Meropenem/vaborbactam,Vabomere
Target:
Carindacillin sodium
Cat.No: T40295
Synonym: Carindacillin sodium,CP-15464-2,Carbenicillin indanyl sodium
Target:
Talampicillin
Cat.No: T34776
Synonym:
Target:
Nitrofurantoin-13C3
Cat.No: T36537
Synonym: Nitrofurantoin-13C3
Target:
Trimethoprim hydrochloride
Cat.No: T75291
Synonym:
Target:
Flumequine-13C3
Cat.No: T36021
Synonym: Flumequine-13C3
Target:
Pazufloxacin
Cat.No: T75296
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T9599 3,4,5-Trimethoxybenzaldehyde

Anti-infection; Antibacterial Microbiology/Virology
3,4,5-Trimethoxybenzaldehyde 是合成各种药物,特别是治疗细菌感染的甲氧苄啶的中间体,它有抗念珠菌功效并抑制粘附和生物膜。
T1313 Nitrofurantoin

Furadantine,呋喃妥因,Macrodantin,Furadonine

Antibacterial; Antibiotic Microbiology/Virology
Nitrofurantoin (Furadantine) 是一种具有口服活性的广谱内酰胺酶抗菌剂。它是一种抗生素,可研究尿路感染。
T4816 6-Hydroxynicotinic acid

6-Hydroxypyridine-3-carboxylic acid,6-羟基烟酸,2-Hydroxy-5-pyridinecarboxylic acid

Others; Endogenous Metabolite Metabolism; Others
6-Hydroxynicotinic acid (6-Hydroxypyridine-3-carboxylic acid) 用于核磁共振波谱或气相色谱-质谱法诊断尿路感染中的铜绿假单胞菌。在引起尿液感染的常见细菌中,只有铜绿假单胞菌从烟酸中产生6-羟基烟酸。

天然产物

3,4,5-Trimethoxybenzaldehyde
Cat.No: T9599
Synonym:
Target: Anti-infection, Antibacterial
Nitrofurantoin
Cat.No: T1313
Synonym: Furadantine,呋喃妥因,Macrodantin,Furadonine
Target: Antibacterial, Antibiotic
6-Hydroxynicotinic acid
Cat.No: T4816
Synonym: 6-Hydroxypyridine-3-carboxylic acid,6-羟基烟酸,2-Hydroxy-5-pyridinecarboxylic acid
Target: Others, Endogenous Metabolite
TargetMol Loading
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